论文部分内容阅读
Design and synthesis of indoline thiohydantoin derivatives based on enzalutamide as antiproliferativ
【机 构】
:
Department of Medicinal Chemistry, China Pharmaceutical University, 24 Tongjiaxiang, Nanjing 210009,
【出 处】
:
2016年长三角药物化学研讨会
【发表日期】
:
2016年11期
其他文献
Design, Synthesis, and Evaluation of Asymmetric EF24 Analogues as Potential Anti-Cancer Agents for L
The nuclear factor-kappa B (NF-κB) signaling pathway has been targeted for the therapy of various cancers,including lung cancer.EF24 was considered as a potent inhibitor of NF-κB signaling pathway.
Synthesis and Biological Evaluation of 6-fluoro-3-phenyl-7-piperazinyl Quinolone Derivatives as Pote
会议
Potentiation Study of LG-12, A Small Molecule Inhibitor of PAPR-1, to Temozolomide in Vitro and in V
会议
吉西他滨ProTide前药NUC-1031能够减少耐药发生,已进入临床研究。但仍无法避免对正常组织的损伤。本文设计合成了吉西他滨ProTide乏氧靶向前药,期待获得具有肿瘤靶向释放的吉西他滨ProTide前药。