Synthesis of multi-substituted 2-aminopyrroles/pyridines via chemoselective Michael addition/intramo

来源 :2015年全国药物化学学术会议暨第五届中英药物化学学术会议 | 被引量 : 0次 | 上传用户：njcxm

【摘要】

：

Multi-substituted pyrroles and pyridines are important scaffolds in medicinal chemistry and organic chemistry due to their prevalence in numerous natural products and synthetic compounds.

【作者】

：

Xueyu Qi Haoyue Xiang Qian He and Chunhao Yang

【机构】

：

State Key Laboratory of Drug Research,Shanghai Institute of Materia Medica,Chinese Academy of Scienc

【出处】

：

2015年全国药物化学学术会议暨第五届中英药物化学学术会议

【发表日期】

：

2015年3期

【关键词】

：

aminopyrroles aminopyridines cyclization reaction

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　　Multi-substituted pyrroles and pyridines are important scaffolds in medicinal chemistry and organic chemistry due to their prevalence in numerous natural products and synthetic compounds.

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