One-step Synthesis of Indoloazocines via Gold-Catalyzed Reaction of Indole Functionality with Intern

来源 :The 24th International Society of Heterocyclic Chemistry Con | 被引量 : 0次 | 上传用户:sncyk
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A variety of indoloazocines can be readily prepared by 8-endo-dig cyclization of alkynylindole substrates and following rearrangement by catalysis of Ph3PAuNTf2 or other gold complexes.The reaction conditions are exceptionally mild, and a range of functional groups are easily tolerated.
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