Building Blocks Enabled Drug Discovery (Selected Slides)

来源 :亚太药物研发领袖峰会(Asia Pharma R&D Leaders Summit 2018) | 被引量 : 0次 | 上传用户:cxz2004
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  --An introduction to a catalog of 30,000 plus novel building blocks, which are designed by analysis of the structures of a large number of real marketed and investigational medicines, as well as findings reported in most current literature in medicinal chemistry.--How these building blocks can accelerate the exploration of structure-activity and structure-property relationships in drug discovery.Real cases on solving issues like hERG, improving metabolic stability,increasing solubility, and extending potential patent space, will be discussed.
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