【摘 要】
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The regioselective and diastereoselective allylic amination of allylic polybenzyl ethers using ehlorosulfonyl isoeyanate (CSI) are powerful methods for the prep
【机 构】
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SchoolofPharmacy,SungkyunkwanUniversity,Suwon440-746,Korea
【出 处】
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The 24th International Society of Heterocyclic Chemistry Con
论文部分内容阅读
The regioselective and diastereoselective allylic amination of allylic polybenzyl ethers using ehlorosulfonyl isoeyanate (CSI) are powerful methods for the preparation of α-amino-β-hydroxy acids and five or six-membered heteroeyele compounds.These reactions have been used as key transformations for the syntheses of natural products such as (-)-lentiginosine, DAB, DGDP, deoxoprosophylline and deoxynojirimycin analogues.
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