Sodium Methylate Catalyzed Michael/Cyclization Cascade Reactions of 3-Aminooxindoles with β,γ-Unsatu

来源 :河南省化学会2016年学术年会 | 被引量 : 0次 | 上传用户:bohaiyifan
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  Spirooxindoles are attractive heterocyclic skeletons with broad and promising activities in various therapeutic fields.[1] As this frameworks have existed in a variety of natural products and pharmaceutical lead compounds,which exhibit important biological activities,[2] a lot of efforts have been devoted to the construction of this useful structure by synthetic and medicinal chemists over the past decades.
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