Simultaneous determination of ephedrine,pseudoephedrine and methylephedrine in plasma by LC-MS/MS an

来源 :世界中医药学会联合会方药量效研究专业委员会成立大会暨第二届国际方药量效关系与合理应用研讨会 | 被引量 : 0次 | 上传用户:lantaiwin
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  To support the pharmacokinetics study of maxingshigan decoction in the rat, a facile HPLC-MS/MS method was developed and validated for the simultaneous determination of ephedrine, pseudoephedrine and methylephedrine in rat plasma.The analytes were separated on a Polar-RP column (50×2.0 mm, 2.5 μm) and a triple-quadrupole mass spectrometry equipped with an electrospray ionization (ESI) source was applied for detection.The plasma sample was prepared by a simple protein precipitation and the recovery for all analytes was over 90%.The calibration curves were linear over a concentration range of 0.3-480.0 ng/mL for ephedrine, pseudoephedrine, and methylephedrine.The intra-day and inter-day precision was less than 15% and the relative errors (RE) were all within ±15%.The validated method was successfully applied to a pharmacokinetics study after oral administration of maxingshigang decoction to the rats.
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