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雷帕霉素是吸水链霉菌产生的三烯大环内酯免疫抑制剂,不溶于水,溶于低级醇等大多数有机溶媒。根据抗生素效价测定的杯碟法,采用纸片法进行雷帕霉素生物效价测定,一、二剂量法测定结果经数理统计符合药典规定要求,雷帕霉素结晶品测定的结果与HPLC一致。
Rapamycin is a triene macrolide immunosuppressant produced by Streptomyces hygroscopicus, insoluble in water and soluble in most organic solvents such as lower alcohols. According to the determination of antibiotic potency cup plate method, using paper method rapamycin biological potency determination, one or two dose determination results by the mathematical statistics in line with the provisions of the Pharmacopoeia, rapamycin crystal product determination results and HPLC Consistent.