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本文根据603的结构特点,合成15个新苯甲酰苯胺衍生物,用改良的氯仿诱发小鼠室性心律失常模型筛选,各化合物都具有不同程度的抗心律失常作用。
In this paper, according to the structural features of 603, 15 new benzanilide derivatives were synthesized and the model of ventricular arrhythmia induced by modified chloroform was screened. All the compounds have different antiarrhythmic effects.