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法莫替丁是一个有效的H_2受体拮抗药,用于治疗胃、十二指肠溃疡等,但由于其水溶性低及在胃液中易水解,故其生物利用度较低,且变异性大。应用环糊精可将此药物分子
Famotidine is a potent H 2 receptor antagonist for the treatment of stomach and duodenal ulcer, but its bioavailability is low and its variability is low due to its low water solubility and its hydrolysis in gastric juice Big. Cyclodextrin can be applied to this drug molecule