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1.含速尿100mg 的安瓿制剂:肾功能不全时给予大剂量速尿有效。对此,在日本也有组织地进行了研究。据认为,速尿的生物学利用率在口服时平均为51%,该利用率因赋形剂不同而发生变化,肾功能不全时降低。大量使用速尿时经静脉给药,但日本的速尿注射剂为20mg/2ml,因而使用不便。最近报告,目前已制成每安瓿含速尿100mg 的注射剂。
1. With furosemide 100mg ampoule preparation: Renal insufficiency given high-dose furosemide effective. In this regard, there are also organized studies in Japan. It is thought that the biological utilization rate of furosemide is 51% on average when orally administered, and the utilization rate varies depending on the excipient and decreases when the renal insufficiency is present. Large-scale use of furosemide intravenously, but Japan’s furosemide injection of 20mg / 2ml, and therefore inconvenient to use. It has recently been reported that injections containing 100 mg of furosemide per ampule have been made so far.