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1981年发表的关于抗肿瘤药物的文章和综述,主要是论述抗肿瘤药物作用机制的新进展。从生物化学方面研究和评价化疗抑制剂的设计和活性,化学致癌的机制和预防及治疗的方法。具有抗肿瘤活性的天然化合物仍然是药物的重要来源和设计新药的依据。。烷化剂新型高效亚硝脉类*)抗小鼠L 1210白血病的疗效比环己亚硝腺(o*m大n4倍。尸一羟基由于分子内环化作用使分子非酶性活化,不产生异氨酸酯。
Published in 1981 on the antitumor drugs articles and reviews, mainly on the mechanism of antitumor drugs new progress. From biochemistry research and evaluation of the design and activity of chemotherapy inhibitors, mechanisms of chemical carcinogenesis and prevention and treatment methods. Natural compounds with antitumor activity remain an important source of drugs and the basis for designing new drugs. . Alkylating agents New high-efficiency nitrosamines *) anti-mouse L 1210 leukemia than the nitrosamine nitric oxide (n * 4 times larger, corpse a hydroxyl due to intramolecular cyclization of non-enzymatic molecule activation, not Isocyanate ester is produced.