LC-MS determination and pharmacokinetic study of salidroside in rat plasma after oral administration

来源 :Journal of Pharmaceutical Analysis | 被引量 : 0次 | 上传用户:zhanranran
下载到本地 , 更方便阅读
声明 : 本文档内容版权归属内容提供方 , 如果您对本文有版权争议 , 可与客服联系进行内容授权或下架
论文部分内容阅读
A simple,rapid and sensitive liquid chromatography-mass spectrometry(LC-MS)method was developed for the determination of salidroside in rat plasma and study of its pharmacokinetics after oral administration of suspension of Erzhi Wan and Fructus Ligustri lucidi into Wistar rats.Plasma sample of 200 μL was extracted with acetic ether-isopropanol(2∶1)and the extraction was performed on a Kromasil C18 column(150 mm×4.6 mm,5 μm)with the mobile phase of methanol-water(41∶59,v/v)within a run time of 6.0 min.The analyte was monitored with positive electrospray ionization(ESI)by selected ion monitoring(SIM)mode.The target ions were m/z 323.05 for salidroside and m/z 411.05 for internal standard(IS)geniposide.A good linear relationship was obtained over the range of 5.0-500.0 ng/mL and the lower limit of quantification was 5.0 ng/mL.The validated method was successfully applied to the pharmacokinetic study of salidroside in rat plasma after oral administration of suspension of Erzhi Wan and Fructus Ligustri lucidi. A simple, rapid and sensitive liquid chromatography-mass spectrometry (LC-MS) method was developed for the determination of salidroside in rat plasma and study of its pharmacokinetics after oral administration of suspension of Erzhi Wan and Fructus Ligustri lucidi into Wistar rats.Plasma sample Of 200 μL was extracted with acetic ether-isopropanol (2:1) and the extraction was performed on a Kromasil C18 column (150 mm×4.6 mm, 5 μm) with the mobile phase of methanol-water (41:59, v/ v) within a run time of 6.0 min. The sample was monitored with positive electrospray ionization (ESI) by selected ion monitoring (SIM) mode. The targetions were m/z 323.05 for salidroside and m/z 411.05 for internal standard (IS )geniposide.A good linear relationship was obtained over the range of 5.0-500.0 ng/mL and the lower limit of quantification was 5.0 ng/mL.The validated method was successfully applied to the pharmacokinetic study of salidroside in rat plasma after oral administration of Suspension of Erzhi Wan And Fructus Ligustri lucidi.
其他文献
我的一位老同学,一天在做常规检查时,被医生检查出胃癌来,只剩下三到六个月的寿命可活。老同学是一个不大不小的行政单位的一把手,年轻有为,作为副处级后备干部已培养两年,刚
2001年该卫生监督所成立以来.经过几年的努力,区、街道、社区(村)三级卫生监督体制建设全面提速。2002年在街道建立了卫生监督分所,并建立了街道卫生检查员队伍,实现了传统监
【目的】探讨中药复方益肾活血解毒汤对实验性动脉粥样硬化(AS)家兔血清炎症标志物的影响及其抗AS的可能作用机制。【方法】将24只青紫蓝兔随机分为2组,空白对照组6只,造模组
在江苏省通州市财政系统,有一个以“老”而出名的人:平日里,上下左右都半开玩笑地称他“张老”;看到他拟定的之件时,大家称他“老笔”;乡村干部见了.称他“老熟人”;在处理
Ring columns placed upstream of a bridge pier to protect it from local scouring are typical scouring countermeasures.A series of experiments are conducted under
《天津市“十二五”时期公路发展规划》《天津市快递服务发展“十二五”规划》《天津市“十二五”时期公路发展规划》至“十二五”期末,天津市高速公路总里程将达到1300公里,
ESPN专栏作家里克·莱利回顾了华裔球星林书豪在成名之前屡次被NCAA和NBA忽视的故事,而那些错过他的名教练们如今追悔莫及。当年,林书豪没能得到任何NCAA一级联盟球队的奖学
国有经济战略重组与国有企业分类改革──如何科学地把握“抓大放小”汪异明(一)1995年中央提出了"抓大放小"的国有经济改革思路,即"抓好大的,放活小的",抓"关键的少数",放一般多数。这一思路
刀耕火种的年代,人类缺少生存的粮食。为了争夺粮食资源,部落之间以及后来的国与国之间发生过无数次大大小小的战争。  农业生产落后的时期,人类缺粮。农业生产发达的今天,人类也还是会时不时地缺少粮食。联合国农业署的一项重要任务,就是逐步减少世界上的饥饿人口。  地球的陆地面积虽然不小,但是山地、沙漠占有很大比例,很多地区是不适合种植粮食的。地球上适合种植粮食的肥沃土地本来就不多,多数集中在沿海沿河的平原
60多岁的黎和亮是湛江市劳动学会副会长(正处级离休干部),近两年来,他以“只争朝夕”的精神,在劳动学会的发展上,倾洒了无数的汗水和心血。1992年3月份,市企业三项劳动制度