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本文首次报道了一个全新吡喃酮香豆素化合物6的合成,经过结构分析确定为天然产物海棠果素(红厚壳烯酮内酯,calophyllolide)的类似物;并对其进行了初步抗炎活性研究,结果表明该化合物对角叉菜胶导致的大鼠踝关节水肿有明显的抑制作用。
This paper reports for the first time the synthesis of a new pyrantel coumarin compound 6, which was identified as a structural analogue of the natural product calophyllolide by structural analysis; and preliminary anti-inflammatory Activity studies, the results show that the compound on carrageenan-induced rat ankle joint edema significantly inhibited.