The authors thank the 100 Talents program of Chinese Academy of Sciences, the Chengdu Institute of 0rganic Chemistry, and the Graduate School of the Chinese Academy of Sciences for financial support o
Twenty-three 1 -(1H-1,2,4-triazole-1 -y1)-2-(2,4-difluorophenyl)-3-(iV-cycloproyl-N-substituted-amino)-2-propanols were designed and synthesized on the basis of