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1972年Singh和Vaughan Willians发现钙拮抗剂的原型维拉帕米的电生理特性明显不同于β-肾上腺素能阻滞剂以及局部麻醉型抗心律失常药物(如奎尼丁).钙拮抗剂
Singh and Vaughan Willians in 1972 found that the electrophysiological properties of the prototype calcium antagonist verapamil were significantly different from those of β-adrenergic blockers and topical anesthetic antiarrhythmic drugs such as quinidine