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作者合成了一系列N′-(2-恶唑基咪基)磺胺类化合物。其合成路线及化合物如下:这些化合物保持了磺胺脒有效的氨基,在体内很少吸收,其中以
The authors synthesized a series of N ’- (2-oxazolylimino) sulfonamides. The synthetic routes and compounds are as follows: These compounds retain the effective amino group of sulfanilamide, which is rarely absorbed in the body,