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【化学名】 4-(1,2∶5,6-二苯并环庚三烯叉)-1-甲基哌啶盐酸盐【结构式】【作用特点】本品为组织胺H:受体拮抗剂,是一种新型的治疗消化性溃疡药物。它能有效地抑制基础胃酸分泌,而且对组织胺、五肤胃泌素等刺激的胃酸分泌也具有明显的抑制作用。单次口服300毫克,可使基础胃酸分泌降低到零。本品口服吸收迅速,半小时内显效,2小时作用可达最高峰,作用可持续3一6小时。本品用于治疗胃及十二指肠溃疡,幽门前溃疡,可使症状迅速消除,对十二指肠溃疡疗效尤为显著。但停药后易复发。【适应症】主治十二指肠溃疡和胃溃疡,也可用于治疗急性胃粘膜出血、胰源性溃疡综合症等。
【Chemical Name】 4- (1,2: 5,6-dibenzocycloheptene) -1-methylpiperidine hydrochloride 【Structure】 【Features】 This product is histamine H: receptor Antagonists, is a new type of drug for treating peptic ulcer. It can effectively inhibit the basic gastric acid secretion, but also on histamine, five gastrin stimulated gastric acid secretion also has a significant inhibitory effect. A single oral 300 mg, can reduce the basic gastric acid secretion to zero. This product oral absorption quickly, markedly within half an hour, up to 2 hours the role of peak, the role of sustainable 3 to 6 hours. This product is used to treat stomach and duodenal ulcer, pyloric ulcer, can quickly eliminate the symptoms, especially for duodenal ulcer. However, easy to relapse after stopping. Indications Indications duodenal ulcer and gastric ulcer, can also be used to treat acute gastric mucosal hemorrhage, pancreatic ulcer syndrome.