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报道了肾显像剂99mTc-1,2-二羟基丙基磷酸(Diol)的制备方法及其动物实验研究。结果显示,99mTc-Diol注入小鼠体内5min后在肾脏达最大摄取率(34.06±4.67%ID/g);注入家兔5min后双肾动态显像最清晰。表明99mTc-Diol是一种肾脏摄取率高、摄取速度快的新型肾显像剂。
The preparation of 99mTc-1,2-dihydroxypropylphosphoric acid (Diol) and its animal experiment were reported. The results showed that the maximal uptake rate of 99mTc-Diol in the kidneys was 34.06 ± 4.67% ID / g after being injected into the mice for 5min. 99mTc-Diol is a new kidney imaging agent with high uptake rate and fast uptake rate.