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酮康唑为咪唑类抗真菌药,对皮肤真菌、酵母菌和一些深部真菌有效。据临床需要,我们研制成水包油型乳膏,用于治疗体癣、股癣、手足癣、汗斑等皮肤病,取得较为满意疗效。 1 仪器与试药 UV—8458紫外分光光度计(美国惠普公司),酮康唑标准品及原料由南京第二制药厂提供,其它辅料均为药用规格,化学试剂为分析纯。 2 处方与制备 2.1 处方:酮康唑20g,白凡士林50g,单硬酸甘油脂40g,硬脂酸120g,液体石蜡60ml,三乙醇胺1Oml,甘油50ml,羟苯乙酯1g,亚硫酸氢钠1g,维生素E5g,蒸馏水加至1000g。
Ketoconazole is an imidazole antifungal that is effective against dermatophytes, yeasts and some deep fungi. According to clinical needs, we developed an oil-in-water cream for the treatment of body ringworm, jock itch, hand, foot and ringworm, sweat stains and other skin diseases, to obtain more satisfactory results. 1 instruments and reagents UV-8458 UV spectrophotometer (Hewlett-Packard, the United States), ketoconazole standard materials and raw materials provided by the Nanjing Second Pharmaceutical Factory, and other accessories are pharmaceutical specifications, chemical reagents for analytical grade. 2 Prescription and Preparation 2.1 Prescription: ketoconazole 20g, white petrolatum 50g, monoglyceride 40g, stearic acid 120g, liquid paraffin 60ml, triethanolamine 1Oml, glycerol 50ml, hydroxy ethyl 1g, sodium bisulfite 1g , Vitamin E5g, distilled water added to 1000g.