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红霉素是1952年由红霉素链霉菌(Streptomyces erythreus)的培养滤液中得到。由于红霉素对耐青霉素的革兰氏阳性菌具有特别强的抗菌活性,因此在抗生素中占有重要的地位。在临床实践中,通常是在其它抗生素如青霉素治疗无效时才应用的。在治疗严重的急性感染时,特别是需要在血清中造成较高的抗生素浓度时,一般应用它的各种水溶性盐类的注射剂。如磷酸盐、乳糖酸盐、葡庚酸盐等。红霉素的抗坏血酸盐是苏联研制出的红霉素水溶性盐,在苏联已用于临床,据统计
Erythromycin was obtained from the culture filtrate of Streptomyces erythreus in 1952. Because of its strong antibacterial activity against penicillin-resistant Gram-positive bacteria, erythromycin plays an important role in antibiotics. In clinical practice, it is usually applied when other antibiotics such as penicillin are ineffective. In the treatment of severe acute infections, and in particular the need for higher concentrations of antibiotics in the serum, the injectables of various water-soluble salts thereof are generally employed. Such as phosphate, lactobionate, glucoheptanoate and the like. Erythromycin ascorbate is the Soviet Union developed erythromycin water-soluble salts, has been used in clinical medicine in the Soviet Union, according to statistics