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蝙蝠葛苏林碱(daurisoline,Dau)是从防己科植物蝙蝠葛根茎中提取的生物碱,(-)-S·R-Dau是其人工合成非对映异构体.研究表明它的药理活性比天然品强很多[1].我们最近报道(-)-S·R-Dau能抑制谷氨酸(Glu)对原代培养的大鼠皮...
Daucus dauricum (Dau) is an alkaloid extracted from the root tuber of Daphniphyllum, and (-) - S · R-Dau is its synthetic diastereomer. Studies have shown that its pharmacological activity is much stronger than natural products [1]. We recently reported that (-) - S · R-Dau can inhibit glutamate (Glu) on primary cultured rat skin ...