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通过 3步合成了对氟苄胺 ,采用均匀试验设计对合成条件进行了研究。结果显示 ,3步合成对氟苄胺工艺可行 ,均匀试验设计方法可方便快捷地优化出最佳合成工艺 ,最佳温度为 1 38℃。
Fluoro-benzylamine was synthesized in three steps and the synthesis conditions were studied using uniform experimental design. The results showed that the three-step synthesis of fumingbenamine process feasible uniform design method can be easily and quickly optimize the optimal synthesis process, the best temperature of 138 ℃.