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Pharmacophore-based design,synthesis,and biological evaluation of novel 3-((3,4-dichlorophenyl)(4-su
[期刊论文] 作者:Dong-Mei Zhao,Wen-Yan Li,Yu-Fang Shi,Xu-Qiong Xiong,Shuai Song,Chen-Zhou Hao,Mao-Sheng Cheng,Jing-Kang,
来源:Chinese Chemical Letters 年份:2014
Cholesteryl ester transfer protein(CETP) is a plasma glycoprotein that plays an important role in decreasing high-density lipoprotein cholesterol(HDL-C) levels...
[期刊论文] 作者:Hong-Lei Xie,Chun-Chi Liu,Yi-Qun Li,Chang-Lin Bai,Chen-Zhou Hao,Jing Guo,Chang-Qun Luo,Dong-Mei Zhao,,
来源:Chinese Chemical Letters 年份:2017
A novel series of β-propanamide derivatives as inhibitors of cholesteryl ester transfer protein(CETP)were synthesized.Previously,H3(IC_(50) 2 μmol/L) was obse...
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