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,Discovery and structural optimization of 4-(4-(benzyloxy)phenyl)-3,4-dihydropyrimidin-2(1H)-ones as
[期刊论文] 作者:Xi-shan WU,Rui WANG,Yan-li XING,Xiao-qian XUE,Yan ZHANG,Yong-zhi LU,Yu SONG,
来源:中国药理学报(英文版) 年份:2016
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,Y08197 is a novel and selective CBP/EP300 bromodomain inhibitor for the treatment of prostate cance
[期刊论文] 作者:Ling-jiao Zou,Qiu-ping Xiang,Xiao-qian Xue,Cheng Zhang,Chen-chang Li,Chao Wang,Qiu Li,Rui Wang,Shuang,
来源:中国药理学报(英文版) 年份:2019
In advanced prostate cancer,CREB (cAMP-responsive element-binding protein) binding protein (CBP) and its homolog EP300 are highly expressed;targeting the bromod...
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