Pd-catalyzed Cross-Coupling of Benzylboronic Acid Pinacol Ester with 1-tert-Butoxycarbonyl-3-iodoaze

来源 :第十九届全国金属有机化学学术讨论会 | 被引量 : 0次 | 上传用户:mingxingc
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T Azetidine derivatives are one of the most important building blocks in pharmaceutical research.[1] The typical procedure for direct alkylation of azetidines is the Ni-catalyzed or Pd-catalyzed Suzuki cross-coupling of alkyl-9-BBN with alkyl halides.
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