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恩杂鲁胺(enzalutamide)为第二代雄激素受体拮抗剂,由Medivation 公司和Astellas公司合作开发,商品名为Xtandi,用于治疗去势难治性前列腺癌(CRPC)[1,2]。
恩杂鲁胺的合成工艺改进
【摘 要】
：
恩杂鲁胺(enzalutamide)为第二代雄激素受体拮抗剂,由Medivation 公司和Astellas公司合作开发,商品名为Xtandi,用于治疗去势难治性前列腺癌(CRPC)[1,2]。
【机 构】
：
武汉工程大学化工与制药学院,武汉,430074 武汉工程大学绿色化工过程教育部重点实验室,武汉,4
【出 处】
：
2015年全国药物化学学术会议暨第五届中英药物化学学术会议
【发表日期】
：
2015年3期
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