Synthesis and anti-inflammatory activity of imidazo [1,2-a] pyrimidine derivatives

来源 :中国化学快报(英文版) | 被引量 : 0次 | 上传用户:fternally
下载到本地 , 更方便阅读
声明 : 本文档内容版权归属内容提供方 , 如果您对本文有版权争议 , 可与客服联系进行内容授权或下架
论文部分内容阅读
A series of imidazo [1,2-a] pyrimidine derivatives substituted adjacently with two aryls at positions 2 and 3 were designed and synthesized in order to improve their anti-inflammatory activities. Biological tests suggested that these compounds have antiinflammatory activities with COX-2 selectivity to some extent.
其他文献
Histone deacetylases (HDACs) play an important role in tumorigenesis. Inhibition of HDACs is considered as a potent strategy for cancer therapy. Two lead compou
The interaction ofbromothymol blue(BB) with human serum albumin(HSA) was studied by electrochemical techniques and a sensitive method for proteins assay was dev
One new (Sarsasapogenin O) and seven known steroids were isolated from the roots of Asparagus officinalis L. Their structures were elucidated on the basis of sp
In this work, the preparation of α, ω-dichloride-terminated multi-vinyl branched siloxane 1 (yield: 57.1%) used for self-healing polymer composites were synth
The Riemann problems for the Euler system of conservation laws of energy and momentum in special relativity as pressure vanishes are considered. The Riemann sol
The fractionated crystallization behavior of the minor dispersed HDPE phase in PS/POE/HDPE/SBS quaternaryblends was investigated by differential scanning calori
The title compound α,α'-bis(3,5-bismethyl-pyrozole-N-yl)-carbene-acetyl-isopro-penyl hydrazine (C16H22N6O, Mr = 314.40) has been prepared. It was characterize
The mixing of particulates such as powders is an important process in many industries including pharmaceuticals, plastics, household products (such as detergent
The lattice Boltzmann method was used to investigate numerically the fiber orientation distributions in slit channel flows with abrupt expansion for fiber suspe
The authors consider a differentiable manifold with Ⅱ-structure which is an isomorphic representation of an associative, commutative and unitial algebra. For R