Synthesis and Bioactivity of Natural Occurring Petasin-Like Derivatives as Antitumor Agents

来源 :药物化学期刊(英文) | 被引量 : 0次 | 上传用户:jing4912
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Petasin is a potential antitumor against human neuroblastoma cell SK-N-SH by inhibiting the ERK1/2 phosphorylation. In view of its great activity and new antiproliferative mechanisms, a series of petasin derivatives were designed and synthesized, which sh
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