The Synthesis of Some 17-(2'-Oxazolyl)-androsta-5,16-diene Deriva-tives as 17α-Hydroxylase/C17,20 -L

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Several 4'- and 5'-substituted 17-(2'-oxazolyl)-androsta-5,16-diene derivatives were designed and synthesized as inhibitors of 17α-hydroxylase/C17,20 -Lyase (P45017α) for the treatment of prostatic cancer, the results of the preliminary pharma
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