2. 您的位置
3. 首页
4. 会议论文
5. One-pot Synthesis of 3,4-Dihydropyridin-2-ones via Tandem Reaction of Blaise Reaction Intermediate a

One-pot Synthesis of 3,4-Dihydropyridin-2-ones via Tandem Reaction of Blaise Reaction Intermediate a

来源 :中国化学会第九届全国有机化学学术会议 | 被引量 : 0次 | 上传用户：maotian1

【摘 要】

：

3,4-Dihydropyridin-2-ones are embedded as a prominent substructure in numerous bioactive compounds exhibiting various activities such as antibacterial,1 antifungal2 and antitumor,3 also served as kina

【作 者】

：

Tuanjie Meng Lantao Liu Cuilan Feng Xiaojuan Wang Wenxian Zhao 

【机 构】

：

College of Chemistry and Chemical Engineering,Shangqiu Normal University,Shangqiu 476000

【出 处】

：

中国化学会第九届全国有机化学学术会议

【发表日期】

：

2015年7期

下载到本地 , 更方便阅读

下载此文 赞助VIP

声明 : 本文档内容版权归属内容提供方 , 如果您对本文有版权争议 , 可与客服联系进行内容授权或下架

论文部分内容阅读

3,4-Dihydropyridin-2-ones are embedded as a prominent substructure in numerous bioactive compounds exhibiting various activities such as antibacterial,1 antifungal2 and antitumor,3 also served as kinase inhibitors.

其他文献

两种二取代四唑异构体的鉴别及其热性能研究

四唑作为富氮杂环化合物,在制药1、含能材料2、多孔材料3 以及燃料4 等方面具有广泛的研究及使用价值.然而,由于四唑二取代化合物具有1,5-二取代和2,5-二取代两种取代类型,在制备四唑高分子及其他四唑衍生物的过程中,常常会因四唑取代类型的不同而生成多种产物,为其分离纯化带来了很大的不便.

会议

Transition-Metal-Free Persulfuration to Construct Unsymmetrical Disulfides and Mechanistic Study of

Our study focused on building C-S,and S-S bonds by using inorganic sulfide agents such as Na2S2O31and RSO2Na.

会议

铜促进的C(sp3)-H键叠氮化反应用于含氮杂环的合成

含氮杂环广泛存在于天然产物,药物,材料分子中,因而,它们的合成方法一直备受化学家们的关注[1].近年来,随着过渡金属催化的C-H 键活化反应的快速发展,通过对分子内的C-H 键直接胺化或酰胺化反应来构建C-N 键正逐渐成为更加有效的含氮杂环的合成策略.

会议

Cascade Synthesis of Spirooxindole δ-Lactone Derivatives through N-Aryl hydroxymethylacrylamides wit

The spirooxindoles are among the most privileged scaffolds in medicinal chemistry.

会议

安宫黄体酮绿色合成技术的研究与应用

安宫黄体酮(Medroxy progesterone acetate)俗称甲孕酮、甲羟孕酮，药名：醋酸甲羟孕酮酸酯、醋酸甲羟孕酮，临床上是甾体孕激素类药，无雌激素活性，孕激素活性在皮下注射为黄体酮的20～30 倍，有长效性。研究表明，安宫黄体酮还具有抗癌活性，用于晚期乳腺癌、子宫内膜癌治疗[1]，和化疗药物合用，效果明显提高，已用于临床，其需求前景广阔，探索绿色合成安宫黄体酮新技术迫在眉梢。

会议

安宫黄体酮甾体药物中间体绿色合成结构表征

Synthesis of 1H-Pyrazolo[4,3-c]quinolines and 4-Anilinoquinoline-3-carbonitriles from 4-Chloroquinol

Quinolines are "privileged" moieties in medicinal chemistry research.

会议

微波辅助合成嘌呤二磷酸

嘌呤二磷酸化合物是近年发现的一种潜在抗骨质疏松化合物[1].传统合成方法,以腺嘌呤为起始原料,采取加热回流的方式,经过N-烃化反应、水解以及二磷酸化反应,得到最终产物.

会议

A Strategy for 2,3-Disubstituted Quinolines Synthesis via Palladium-Catalyzed Oxidative C-C bond Cle

As powerful strategies to construct multiple carbon-carbon and carbon-heteroatom bonds,palladium-catalyzed effective transformations of alkenes and alkynes have attracted increasing attention in the p

会议

Synthesis of Fullerene-Fused Dioxygenated Ring Compounds:TsOH-Mediated Novel Reaction of Aziridinofu

Chemical modification of fullerenes to produce fullerene derivatives with one or several addends covalently bound to the spherical carbon framework have attracted extensive attention in the chemical c

会议

Ferric Perchlorate-Mediated One-Step Reaction of [60]Fullerene with Diols for the Preparation of Ful

Many chemical reactions have been discovered over the past two decades,and a large number of fullerene derivatives with widely structural diversities have been prepared.

会议