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5. Asymmetric Synthesis of Tetrahydro-β-carbolines via Chiral Phosphoric Acid Catalyzed Transfer Hydrog

Asymmetric Synthesis of Tetrahydro-β-carbolines via Chiral Phosphoric Acid Catalyzed Transfer Hydrog

来源 :The 24th International Society of Heterocyclic Chemistry Con | 被引量 : 0次 | 上传用户：cheney0105

【摘 要】

：

An efficient synthesis of enantioenriched tetrahydro-β-carbolines via chiral phosphoric acid catalyzed enantioselective transfer hydrogenation of hydroxylactams has been achieved.This methodology feat

【作 者】

：

Qin Yin Shu-Li You 

【机 构】

：

State Key Laboratory of Organometallic Chemistry,Shanghai Institute of Organic Chemistry,Chinese Aca

【出 处】

：

The 24th International Society of Heterocyclic Chemistry Con

【发表日期】

：

2013年4期

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论文部分内容阅读

An efficient synthesis of enantioenriched tetrahydro-β-carbolines via chiral phosphoric acid catalyzed enantioselective transfer hydrogenation of hydroxylactams has been achieved.This methodology features the ready availability of the starting materials, high yields, and mild reaction conditions.

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