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5. PIFA-Mediated Oxidation of β-Ketoamide:Synthesis of vicinal tricarbonyl Amides

PIFA-Mediated Oxidation of β-Ketoamide:Synthesis of vicinal tricarbonyl Amides

来源 :河南省化学会2016年学术年会 | 被引量 : 0次 | 上传用户：davidrandy

【摘 要】

：

A facile and direct synthetic method for the synthesis of vicinal tricarbonyl amides(VTAs)in moderate to excellent yields(62-93%)has been developed starting from readily available β-ketoamide in the p

【作 者】

：

Yueyang Liu Yameng Wan Zhiguo Zhang Guisheng Zhang 

【机 构】

：

Collaborative Innovation Center of Henan Province for Green Manufacturing of Fine Chemicals,Key Labo

【出 处】

：

河南省化学会2016年学术年会

【发表日期】

：

2016年10期

【关键词】

：

Vicinal tricarbonyl amides (VTAs) vic-Diketoamides β-Dicarbonyl compounds β-Keto 

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论文部分内容阅读

　　A facile and direct synthetic method for the synthesis of vicinal tricarbonyl amides(VTAs)in moderate to excellent yields(62-93%)has been developed starting from readily available β-ketoamide in the presence of sole phenyliodine(Ⅲ)bis(trifluoroacetate)(PIFA).

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