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5. Diversity-oriented Synthesis of 2-Substituted Purine Nucleosides from Readily Available Starting Mat

Diversity-oriented Synthesis of 2-Substituted Purine Nucleosides from Readily Available Starting Mat

来源 :河南省化学会2016年学术年会 | 被引量 : 0次 | 上传用户：lingdujimo

【摘 要】

：

2-substituted purine nucleosides have received considerable attention due to their broad spectrum of biological activities.Thus,numerous economically important pharmaceuticals,such as cladribine,Regad

【作 者】

：

Xi-Ning Yang Ran Xia Gui-Rong Qu 

【机 构】

：

College of Chemistry and Chemical Engineering,Henan Normal University,Xinxiang,P.R.China,453007

【出 处】

：

河南省化学会2016年学术年会

【发表日期】

：

2016年10期

【关键词】

：

diversity-oriented synthesis 2-substituted purine nucleosides late-stage nitrati 

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论文部分内容阅读

　　2-substituted purine nucleosides have received considerable attention due to their broad spectrum of biological activities.Thus,numerous economically important pharmaceuticals,such as cladribine,Regadenoson,fludarabine,Cangrelor or nelarabine,have 2-substituted purine units as indispensable substructures.

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