【摘 要】
:
2,3-Dihydrobenzofurans are unique structural skeletons in many biologically active molecules and natural products.An atom economical method for the synthesis of 2,3-dihydrobenzofurans via the o-QMs ge
【机 构】
:
State Key Laboratory of Catalysis,Dalian Institute of Chemical Physics,Chinese Academy of Sciences,4
【出 处】
:
The 24th International Society of Heterocyclic Chemistry Con
论文部分内容阅读
2,3-Dihydrobenzofurans are unique structural skeletons in many biologically active molecules and natural products.An atom economical method for the synthesis of 2,3-dihydrobenzofurans via the o-QMs generated from readily available 2-alkylsubstituted phenols using Ag2O mediated oxidation has been developed.This methodology provides a facile access to 2,3-dihydrobenzofurans in moderate to good yields and excellent diastereoselectivity.
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