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本品为抗高血压药,化学名为N-脒基-2-(2,6-二氯苯基)乙酰胺盐酸盐。药理本品对于患原发性高血压、DO-CA高血压、肾性高血压的大白鼠及患Gold-blatt高血压的狗在麻醉和非麻醉条件下给药的研究表明,其降压作用相当于氯压定的十分之一。本品无氯压定的反跳现象,困倦、口渴等副作用也比氯压定弱。其作用机理和氯压定相同,均为对中枢神经系统的肾上腺素α受体的直接刺激作用,但作用点的细节方
This product is anti-hypertensive drugs, chemical name for the N-amidino-2- (2,6-dichlorophenyl) acetamide hydrochloride. Pharmacology This product is administered to anesthetized and non-anesthetized rats in hypertensive rats with essential hypertension, DO-CA hypertension, and renal hypertension and dogs with Gold-blatt hypertension, indicating that its antihypertensive effect Equivalent to chlorine pressure set one-tenth. This product chlorine-free pressure rebound phenomenon, drowsiness, thirst and other side effects than chlorine pressure set weak. Its mechanism of action and chlorine pressure set the same, are on the central nervous system adrenaline α receptor stimulation, but the details of the role of points