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Inordertostudytherelationsbetweenstructureandactivityandfoundmorepotentialallostericmodulatorofmuscarinicm2-receptor,aseriesofW84analogouswithpiperazinyldithiocarbonateweredesignedandsynthesizedbasedonthestructureofW84[1]andthenewsyntheticmethodofdithioca
Inordertostudytherelationsbetweenstructureandactivityandfoundmorepotentialallostericmodulatorofmuscarinicm2-receptor, aseriesofW84alogouswithiperazinyldithiocarbonateweredesignedandsynthesizedbasedonthestructureofW84 [1] and the newsyntheticmethodofdithioca