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秦艽生物碱甲为自中药秦艽根提出的一种生物碱.给大鼠腹腔注射秦艽生物碱甲180及250毫克/公斤,能使血糖升高.此作用在给药后半小时即出现,维持约3小时.秦艽生物碱甲150-250毫克/公斤亦能引起小鼠血糖升高,剂量愈大作用愈强.动物切除肾上腺后再注射秦艽生物碱甲,则不复出现血糖的升高。在秦艽生物碱甲升高血糖的同时,盰糖元明显降低.肾上腺素能阻断药能部分或完全阻断秦艽生物碱甲的作用。以上结果说明秦艽生物碱甲具有升血糖的作用,此作用可能主要系通过肾上腺素的释放.
Gentiana straminea alkaloid is a kind of alkaloid proposed from Gentiana straminea.Animals injected intraperitoneally with Gentiana macrophylla 180 and 250 mg / kg, can make blood sugar rise.This effect appears half an hour after administration, maintain About 3 hours.Alcanthinol 150-250 mg / kg also can cause mice to rise in blood sugar, the greater the role of the stronger the dose.After removal of the animal adrenalectin injection of Qin Fang alkaloid A, no increase in blood sugar. In the Qionglai alkaloids A blood sugar increased at the same time, 盰 glycogen significantly reduced.Adrenergic blocking drugs can partially or completely block the role of Qin Fang alkaloids. The above results show that Qin Jia alkaloid A has the role of blood glucose, this effect may be mainly through the release of epinephrine.