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目的:介绍微透析采样技术在抗乳腺癌药物方面的研究与应用现状。方法:参阅国内外文献,进行分析、归纳和总结。结果:微透析采样技术在乳腺癌的发病机制、乳腺癌药物临床前和临床药理及药动学、PK-PD结合模型、联合用药合理性等方面研究应用广泛。结论:微透析采样技术结合现代成像技术,在乳腺癌肿瘤局部药动学研究方面具有广阔的应用前景。
Objective: To introduce the status of research and application of microdialysis sampling technology in anti-breast cancer drugs. Methods: Refer to the literature at home and abroad, analyze, summarize and summarize. Results: The microdialysis sampling technique has been widely used in the pathogenesis of breast cancer, preclinical and clinical pharmacology and pharmacokinetics of breast cancer drugs, PK-PD binding model and rationality of combination therapy. Conclusion: The microdialysis sampling technique combined with modern imaging technique has broad application prospects in the study of local pharmacokinetics of breast cancer.