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Azimexone化学名为2-[2-氰氮丙啶基-(1)]2-[2-甲氨酰氮丙啶基-(1)-丙烷;Ciamexone化学名为2-氰基-1-[(2-甲氧基-6-甲基吡啶基-3)甲基]氮丙啶。同属氮丙啶类小分子免疫调节剂。 合成Azimexone的关键是制得2-氰氮丙啶中间体,Schmitz VE报道由环已酮、氢氧化铵
Azimexone has the chemical name 2- [2- cyanopyridyl- (1)] 2- [2-carbamimidazinyl- (1) (2-methoxy-6-methylpyridyl-3) methyl] aziridine. Both belong to the aziridine small molecule immunomodulator. The key to the synthesis of Azimexone is the preparation of 2-cyanopyridine intermediate, Schmitz VE reported by cyclohexanone, ammonium hydroxide