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omapatrilat是布迈-施贵宝(BMS)公司正在开发的治疗高血压和心衰的新产品,为第一个新一类血管肽酶抑制剂,是一种对血管紧张素转化酶(ACE)和中性内肽酶(NEP)起双重抑制作用的单分子物质。ACE可将血管紧张素Ⅰ转化为血管紧张素Ⅱ,血管紧张素Ⅱ
omapatrilat is a new product under development for the treatment of hypertension and heart failure by the Bamy-Bristol-Myers Squibb (BMS) company. It is the first new class of vasopeptidase inhibitors, an inhibitor of angiotensin-converting enzyme (ACE) and Sexual endopeptidase (NEP) plays a dual inhibitory effect of single-molecule substances. ACE can convert angiotensin Ⅰ into angiotensin Ⅱ and angiotensin Ⅱ