论文部分内容阅读
本文报道新颖的6-连氮和6α-甲氧基-6β-取代腙青霉素的合成及引入6α-甲氧基的新方法。这类化合物对一些阴性菌和阳性菌有中等活力,且引入6α-甲氧基之后对细菌的抑制作用增强。
This paper reports the novel synthesis of 6-azin and 6α-methoxy-6β-substituted hydrazone penicillin and a new method of introducing 6α-methoxy. These compounds are moderately active against some of the negative and positive bacteria, and their inhibitory effect on bacteria is enhanced by the introduction of 6α-methoxy.