论文部分内容阅读
目前美国市场上出售的非甾体抗炎药除阿司匹林外,尚有苯氧苯丙酸(fenoprofen)、布洛芬、消炎痛、甲氯灭酸钠、甲灭酸、甲氧萘丙酸(naproxen)及其钠盐、保太松、氧苯保太松、炎痛喜康、苏灵大(sulindac)、托灭停(tolmetin)和佐美酸(zome-ptrac)等。在肝毒性方面:除保太松可能发生肉芽肿肝炎、广泛性肝坏死外,苏灵大、消炎痛、布洛芬、甲氧萘丙酸也可见到胆汁郁积性肝炎、血清转氨酶特别是丙氨酸转氨酶活性在给药头几周后增加,如活性水平超过正常水平上限的3倍则必须停药,药物停用后症状可得到改善。长期使用一种非甾体抗炎药可造成慢性肝炎。
At present, non-steroidal anti-inflammatory drugs sold on the U.S. market include aspirin, fenoprofen, ibuprofen, indomethacin, meclofenamate, mefenamic acid, naproxen naproxen and its sodium salt, loxapine, oxybenzone, piroxicam, sulindac, tolmetin and zome-ptrac and the like. In hepatotoxicity: In addition to Paul too loose may occur granulomatous hepatitis, extensive liver necrosis, Su Ling large, indomethacin, ibuprofen, naproxen can also be found in cholestatic hepatitis, serum transaminases, especially C The aminotransferase activity increases in the first few weeks after administration. If the activity level exceeds the upper limit of normal, it must be discontinued. The symptoms can be improved after the drug is stopped. Long-term use of a non-steroidal anti-inflammatory drugs can cause chronic hepatitis.