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在研究了50 IU/kg(家兔体重)以上剂量的胰岛素栓直肠给药能降低家兔血糖和某些表面活性剂具促进吸收的作用后,本文报导了含有1%表面活性剂 NO—10,剂量为75、50、30、10、5、3 IU/kg 的胰岛素可可豆油栓剂直肠给药后家兔的血糖变化。研究结果表明,75 IU/kg 和50IU/kg 剂量的胰岛素栓能使家兔产生抽搐甚至死亡,30和10IU/kg 的剂量也导致动物在实验期间内(6.0hr)血糖不能回升,5IU/kg 的剂量给药2和6小时后可使家兔血糖分别下降79%和33%。3 IU/kg 剂量的胰岛素栓在给药1.5和6.0小时时使家兔血搪分别下降65%和24%,与对照组相比,作用非常显著(P<0.001)。
After investigating the effects of insulin suppositories at doses above 50 IU / kg (rabbit body weight), which reduce blood glucose levels in rabbits and promote the uptake by certain surfactants, the paper reports the effects of 1% surfactant NO-10 , The dose of 75,50,30,10,5,3 IU / kg of insulin cocoa butter suppository after rectal blood glucose changes in rabbits. The results showed that 75 IU / kg and 50 IU / kg of insulin suppository produced convulsions and even death in rabbits. The doses of 30 and 10 IU / kg also caused the animals to not recover blood glucose during the experimental period (6.0 hr), while 5 IU / kg The blood glucose of rabbits decreased by 79% and 33% respectively after 2 and 6 hours. Insulin suppository at a dose of 3 IU / kg decreased blood viscosity in rabbits by 65% and 24% at 1.5 and 6.0 hours, respectively, which was significantly (P <0.001) comparable to the control group.