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云南白药总皂甙皮下注射,对大鼠佐剂性多关节炎原发病变(35mg/kg×2),角叉菜胶性足肿胀(15,7.5mg/kg),白细胞游走反应(15mg/kg)和棉球肉芽肿(7.5mg/kg/日×7日)均有抑制作用。抗炎机理一部分系通过抑制组胺和PG的释放及对抗其所引起的关节肿胀和毛细血管渗透性增强;另一部分则可能是通过肾上腺皮质系统产生。
Total injection of Yunnanbaiyao saponin subcutaneously on primary lesions of adjuvant-induced polyarthritis in rats (35 mg/kg×2), carrageenan foot swelling (15,7.5 mg/kg), leukocyte migration response (15 mg/ Kg) and cotton ball granuloma (7.5 mg/kg/day x 7 days) all had inhibitory effects. Part of the anti-inflammatory mechanism is through the inhibition of the release of histamine and PG and its resistance to joint swelling and increased capillary permeability; the other part may be through the adrenocortical system.