triazoles相关论文
A Metal-free Multicomponent Cascade Reaction for the Regiospecific Synthesis of 1,5-Disubstituted 1,
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Sterioselective Synthesis of an Important Triazole Intermediate for Antifungal Drugs and its Biologi
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Rhodium(Ⅱ)-Catalyzed [4+3] Cyclization of Triazoles with Indole Derivatives and Its Application in t
Main observation and conclusionrnAn efficient rhodium(Ⅱ)-catalyzed [4+3] cyclization reaction of 1-sulfonyl-1,2-3-triaz......
Over the past few decades,theres an explosive increase of interest in electrophilic cyclization to synthesize carboc......
目的 探讨非艾滋病(AIDS)相关隐球菌性脑膜炎合并脑神经损伤患者的危险因素及预后因素.方法 回顾性分析非AIDS相关隐球菌性脑膜炎1......
A facile and efficient strategy for the synthesis of 5-aryl-2-(quinolin-2-yl)oxazoles via rhodium-catalyzed formal[3+2]c......
目的 评估2009-2011年杭州地区抗深部真菌感染药的临床应用状况,为临床合理应用抗真菌药提供依据.方法 根据杭州地区25家医院2009......
,Novel ferrocenyl derivatives exert anti-cancer effect in human lung cancer cells in vitro via induc
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,Identification of arylamine N-acetyltransferase inhibitors as an approach towards novel anti-tuberc
New anti-tubercular drugs and drug targets are urgently needed to reduce the time for treatment and also to identify age......
该文从挂篮荷载计算、施工流程、支座及临时固结施工、挂篮安装及试验、合拢段施工、模板制作安装、钢筋安装、混凝土的浇筑及养生......
Crystal Structure and DFT Studies of a Triazole Derivative: 4-(2-Hydrobenzylideneamino)-3-(1,2,4-tri
本文通过对荣华二采区10...
Copper Salt of 12-Tungstophosphoric Acid: An Efficient and Reusable Heteropoly Acid for the Click Ch
为探究吕家坨井田地质构造格局,根据钻孔勘探资料,采用分形理论和趋势面分析方法,研究了井田7......
为探究吕家坨井田地质构造格局,根据钻孔勘探资料,采用分形理论和趋势面分析方法,研究了井田7......
Sodium hydride-mediated synthesis of 1,5-diaryl-1,2,3-triazoles from anti-3-aryl-2,3-dibromopropanoi
A series of 1,5-disubstituted 1,2,3-triazoles are synthesized by a one-pot process from anti-3-aryl-2,3-dibromopropanoic......
唑类药物是目前治疗浅部和深部真菌感染的一线用药.按照其结构的不同,该药可以分为咪唑类和三唑类.3种咪唑类新药卢立康唑、拉诺康......
Crystal Structure and DFT Studies of a Triazole Derivative: 4-(2-Hydrobenzylideneamino)-3-(1,2,4-tri
A novel triazole derivative 4-(2-hydrobenzylideneamino)-3-(1,2,4-triazol-4-ylmethyl)-1H-1,2,4-triazole-5(4H)-thione(1) w......
自1999年Barry Sharpless提出点击化学的概念以来，其得到极大的关注和发展。主要介绍了点击化学的定义和分类，其中Cu（I）催化下炔基与叠......
In this paper, the fully optimized molecular geometries and electronic structures of six 1,2,3- and 1,2,4-triazoles were......
A series of novel compounds 3-(2-furyl)-4-aryl-l, 2, 4-triazole-5-thiones have been synthesized. All the compounds were......
本文设计并合成了１０个新的三唑及苯并三唑类化合物，其化学结构均经过有关光谱数据证实，对合成的所有化合物经体外抗真菌试验表明：对所试......
目的：研究１－［２－（取代苯基）－２－（取代苯基甲硫基）乙基］－１Ｈ－１，２，４－三唑类化合物体外抗真菌活性，并初步探讨其构效关系。方法：选择８种临床致病真菌为试验菌，观察本类......
目的 研究一类新型的氮唑化合物对念球菌真菌的抗真菌活性。方法 采用体外抗真菌活性试验，测定化合物的最低抑菌浓度（ＭＩＣ），从而评价化合......
根围土壤稀释培养的结果表明,以R/S为指标,0.03ai.％三唑酮、三唑醇种子处理后,根围引起小麦纹枯病的丝核菌群体明显下降。未进行种......
设计并合成了８个新的三唑及苯并三唑类化合物，其化学结构均经过有关光谱数据证实，对合成的所有化合物经体外抗真菌试验表明；对所试验的......
报道了３９个新的１－｛２－［（取代苯基）甲氧基］－２－（取代苯基）乙基｝－１Ｈ－三唑和苯并三唑类化合物的合成与体外抑菌试验，结果表明，化合物６，１３的抗真菌活性为益康唑的４－１０倍，人......
自1999年Barry Sharpless提出点击化学的概念以来,其得到极大的关注和发展。主要介绍了点击化学的定义和分类,其中Cu（I）催化下炔基与......
目的:研究不同含硫侧链的引入对三唑醇类化合物抗真菌活性的影响.方法:设计合成了15个含硫侧链取代三唑醇类化合物,其中13个为新化......
目的:研究不同取代哌嗪侧链的引入对三唑醇类化合物抗真菌活性的影响.方法:设计合成了11个三唑醇类新化合物;选择8种真菌(白色念珠......
以苯骈三氮唑和氯乙酸乙酯为原料,发生N一烷基化反应,然后再跟水合肼反应制备出苯骈三唑乙酰肼,同时探讨了最佳反应条件,包括反应......
为了提高隐球菌脑膜炎患者脑脊液检测的阳性率，首次使用隐球菌抗原乳胶凝结试验法，对１２例患者进行了检测，阳性率为１００％。该方法快速、敏感和......
[目的]合成具有抗癫痫作用的1-取代苄基-N-环己基-[1,2,3]-三唑-4-甲酰胺衍生物.[方法]采用取代氯苄与叠氮钠反应生成取代苄基叠氮......
Some New Heterocycles from the Reaction of 4-Carboxaldehyde-2-Phenyl-2H-1,2,3-Triazole Malononitrile
Reaction of 4-carboxaldehyde-2-phenyl-2H-1,2,3-triazole 1 with malononitrile in presence of piperidine afforded the tria......
Some New Heterocycles from the Reaction of 4-Carboxaldehyde-2-Phenyl-2H-1,2,3-Triazole Malononitrile
Reaction of 4-carboxaldehyde-2-phenyl-2H-1,2,3-triazole 1 with malononitrile in presence of piperidine afforded the tria......
目的探索合成目标产物1-N和2-N乙腈基取代苯并三氮唑的合成工艺条件。方法以苯并三氮唑和氯乙腈为原料,在不同反应体系（三乙胺/DMF......
目的探讨5-氯苯并三氮唑N-上引入乙腈基所得产物异构体组成分布和产率的影响。方法以5-氯苯并三氮唑和苯并三氮唑分别与氯乙腈反应......
Two new 1,4-disubstituted 1,2,3-triazoles-4-carboxylates were synthesized via click reaction. Compound 1a was synthesize......
从制剂的研发、抗菌性能、抗流失性能、对金属腐蚀性能及生物降解性能等方面介绍了三唑类木材防腐剂的研究进展,对其存在的问题及......
目的：研究地非三唑与黄酮类化合物槲皮素、山奈酚、异鼠李素和四方蒿提取物的代谢相互作用。方法：选取山奈酚、异鼠李素和四方蒿提取......
Reaction of Nitrilimines with 2-Aminopicoline, 3-Amino-1,2,4-Triazole, 5-Aminotetrazole and 2-Aminop
The reaction of picoline derivatives 3-6 with hydrazonoylhalide 1a produced imidazo[1,2-a]pyridines 7-10, while the reac......
In this short review, excerpts from the literature of azo-bridged triazoles(mainly 1,2,4-triazoles), some of their deriv......
Azoniaallene salts as versatile building blocks in the synthesis of antibacterial and antifungal het
Substituted 2-azoniaallene salts 1 are strong bifunctional electrophiles, undergo cyclization reactions furnish many ser......
