Design,synthesis,and biological evaluation of novel class Ⅰ and Ⅱb histone deacetylase inhibitors

来源 :2015年全国药物化学学术会议暨第五届中英药物化学学术会议 | 被引量 : 0次 | 上传用户:ynkm8899
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  Histone deacetylases(HDACs)are a family of enzymes that remove the acetyl groups of acetylated histones or other nonhistone substrates leading to transcriptional repression,and play important roles in the upstream control of chromosome remodeling,gene transcription,cell proliferation and apoptosis.
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