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化学名 (±)5-[1-羟基-2-[[2-(邻甲氧基苯氧基)乙基-]氨基]乙基]-2-甲基苯磺酰胺盐酸盐药效分类抗高血压药开发单位 (日本)山之内制药公司上市厂商 (日本)山之内制药公司,1988年3月29日药理本品对α_1、α_2、β_1、β_2受体的亲和性之间的比约为1∶1/500~1000∶0.3∶0.3。药效为哌唑嗪的1/8~30,普萘洛尔的1/12~16。对各种高血压模型一次给药有迅速而持久的降压效果,耐受性好。
Chemical name (±) 5- [1-hydroxy-2 - [[2- (o-methoxyphenoxy) ethyl] amino] ethyl] -2-methylbenzenesulfonamide hydrochloride Pharmacodynamic classification Antihypertensives Developer (Japan) Yamanouchi Pharmaceutical Co., Ltd. Listed Manufacturer (Japan) Yamanouchi Pharmaceutical Co., Ltd., March 29, 1988 Pharmacological The ratio of the affinity of this product to α_1, α_2, β_1, β_2 receptors is about 1: 1/500 ~ 1000: 0.3: 0.3. Pharmacodynamic prazosin 1/8 ~ 30, propranolol 1/12 ~ 16. A variety of models of hypertension with a rapid and sustained antihypertensive effect, well tolerated.