A Single D-/or L-Isonucleoside Incorporated Thrombin Binding Aptamer

来源 :第九届IUPAC化学生物学国际研讨会暨第八届世界华人药物化学研讨会 | 被引量 : 0次 | 上传用户:cox_7261
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  Thrombin binding aptamer(TBA) is a 15-mer DNA aptamer which was found by SELLEX screening technology.It adopts a chair-type antiparallel G-quartet structure and can specifically interact with thrombin,thus inhibiting blood coagulation of the enzyme activity.Isonucleoside(IsoNA) is a kind of nucleosides whose bases connect to the positions other than C-1 of glycosyl moiety.The local conformation will be changed when IsoNA,especially the L-IsoNA,was incorporated into TBA.
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