青蒿琥酯绿色合成新工艺

来源 :2015年全国药物化学学术会议暨第五届中英药物化学学术会议 | 被引量 : 0次 | 上传用户:aboutt
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  青蒿琥酯(Artesunate 1)是中国首次得到国际承认的独立创制的新药。它是目前世界上最有效的用于治疗脑型疟疾和抗氯喹恶性疟疾的药物。它具有高效、低毒、使用方便、与氯喹无交叉抗药性等特点,经国内外大量临床实验证明,用于治疗各种危重疟疾患者和抢救脑型疟疾病人有很好的疗效。
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